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#3
Le modafinil est un mГ©tabolite actif du R-modafinil et du S-modafinil, ou a fortiori, du mГ©lange racГ©mique du R-modafinil et du S-modafinil. Cet effet serait dГ» Г  un agonisme des rГ©cepteurs de la dopamine D2 et de la sГ©rotonine 5-HT1A. On pense que le modafinil agit sur l'hypothalamus, une partie du cerveau qui contrГґle une grande partie du cycle veille/sommeil.

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Le modafinil ne fonctionne pas non plus pendant la phase de sommeil connue sous le nom de sommeil profond, qui se caractГ©rise par de faibles niveaux de dopamine et de sГ©rotonine. En solution, le Modafinil est extrГЄmement lipophile. Le modafinil est un stimulant oral et agit sur le systГЁme nerveux central en augmentant la dopamine, en inhibant la recapture de la dopamine et en modulant la transmission de la noradrГ©naline. Il est particuliГЁrement indiquГ© pour les travailleurs postГ©s et les personnes souffrant de troubles du sommeil liГ©s au travail postГ©, ainsi que pour les vols long-courriers.
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